PF 3845
发布者:信康 浏览次数:
产品名称:PF 3845CAS:1196109-52-0别名:N-3-吡啶基-4-[[3-[[5-(三氟甲基)-2-吡啶基]氧基]苯基]甲基]-1-哌啶甲酰胺;PF-3845N-3-吡啶-4-[[3-[[5-(三氟甲基)-2-吡啶]氧基]苯基]甲基]-1-哌啶羧酰胺英文名:N-3-Pyridinyl-4-[[3-[[5-(trifluoromethyl)-2-pyridinyl]oxy]phenyl]methyl]-1-piperidinecarboxamide
- 储存条件 Store at +4°C
- 溶解度 DMSO: ≥45mg/mL
- 颜色white to tan
- 用途 PF 3845 is a selective fatty acid amide hydrolase (FAAH) inhibitor (Ki = 0.23 渭M). Reduces inflammatory pain via a cannabinoid receptor-dependent mechanism. Highly efficacious and selective in vivo. Displays no activity at FAAH-2 (IC50 >10 渭M).